Published November 27, 2006
| Accepted Version
Journal Article
Open
The synthesis of C-3β functionalized indoles via a hydroboration/Suzuki–Miyaura coupling sequence
- Creators
- Ferreira, Eric M.
-
Stoltz, Brian M.
Chicago
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Abstract
A method for the functionalization of C-3β of vinyl indoles is described. The procedure involves a hydroboration, followed by a Suzuki–Miyaura cross-coupling with the intermediate alkyl borane. Triflates, bromides, and iodides are suitable coupling partners, allowing access to a variety of elaborated indole compounds.
Additional Information
© 2006 Elsevier Ltd. Received 1 September 2006, Accepted 21 September 2006, Available online 13 October 2006. The authors wish to thank the NIH-NIGMS (R01 GM65961-01), Bristol-Myers Squibb Company (graduate fellowship to E.M.F.), the NSF (graduate fellowship to E.M.F.), the Dreyfus Foundation, Merck Research Laboratories, Research Corporation, Abbott Laboratories, Pfizer, Amgen, GlaxoSmithKline, Lilly, and Johnson and Johnson for their generous financial support.Attached Files
Accepted Version - nihms-13692.pdf
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Additional details
- PMCID
- PMC1832155
- Eprint ID
- 72291
- DOI
- 10.1016/j.tetlet.2006.09.112
- Resolver ID
- CaltechAUTHORS:20161128-080903512
- NIH
- R01GM65961-01
- Bristol-Myers Squibb Company
- NSF
- Camille and Henry Dreyfus Foundation
- Merck Research Laboratories
- Research Corporation
- Abbott Laboratories
- Pfizer
- Amgen
- GlaxoSmithKline
- Lilly
- Johnson and Johnson
- Created
-
2016-11-28Created from EPrint's datestamp field
- Updated
-
2021-11-11Created from EPrint's last_modified field